第 7 章 抗胆碱酯酶药和 胆碱酯酶复活药. 抗 che 药作用原理: che 为 ach...
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7
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(cholinesterase,ChE) ( AChE)ChE
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ChEChEAchChEAch
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, , , ,
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(neostigmine)
AChE.
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1.2.
[]
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1.2.3.
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AchEAchMNN2Ach
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1.2., 3.4.
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MN, ,
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(6~8h)
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1.,,2.
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AchEAchAchM
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1.AchE5~15min 2.
(edrophonium choride)
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2mg30~45 8mg ()
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() ambenonium chloride AchE
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(galanthamine) ()
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(demecarium bromide) AchE15~60min24h19
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DDVPSarin, Tabun
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ChEChEAch,,.
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aging:
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AchE,,AchE,Ach,.
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MNN+
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M,,,,,,
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N,,,
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AChE
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.
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: + : ,
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1. 2. NS2% NaHCO33.
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1. ,,2. ,3.
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cholinesterase reactivatorsPAM PAM-Cl
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PAM
(Oxime), , :ChEPAM
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ChE,
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N>>>>M > , >>>
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1., , , 2.
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M N.
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+ +..
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1.,,2.,,im
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