cheminform abstract: simple and efficient synthesis of belinostat

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ChemInform 2011, 42, issue 01 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim Sulfonamides Q 0560 DOI: 10.1002/chin.201104091 Simple and Efficient Synthesis of Belinostat. — A new route to the potential anti- cancer drug belinostat (VI) is presented. The approach avoids hazardous reagents such as oleum and gives an improved overall yield. — (YANG, L.; XUE*, X.; ZHANG, Y.; Synth. Commun. 40 (2010) 17, 2520-2524, http://dx.doi.org/10.1080/00397910903277870 ; Dep. Med. Chem., China Pharm. Univ., Nanjing 210009, Peop. Rep. China; Eng.) — H. Haber 04- 091

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Page 1: ChemInform Abstract: Simple and Efficient Synthesis of Belinostat

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SulfonamidesQ 0560 DOI: 10.1002/chin.201104091

Simple and Efficient Synthesis of Belinostat. — A new route to the potential anti-cancer drug belinostat (VI) is presented. The approach avoids hazardous reagents such as oleum and gives an improved overall yield. — (YANG, L.; XUE*, X.; ZHANG, Y.; Synth. Commun. 40 (2010) 17, 2520-2524, http://dx.doi.org/10.1080/00397910903277870 ; Dep. Med. Chem., China Pharm. Univ., Nanjing 210009, Peop. Rep. China; Eng.) — H. Haber

04- 091

ChemInform 2011, 42, issue 01 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim

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