2003-2004 gi diseases review 30 november 2015 1:04 am

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2003-2004GI Diseases Review

April 18, 202305:44 PM

Activated charcoal

Antidote

Alosetron

IBS treatment

5HT3 receptor antagonist

Aluminum hydroxide

Antiulcer

Antacid

Amoxicillin

Penicillin antibioticCell wall synthesis inhibitor

Antiulcer

Amino penicillinInhibits peptidoglycan cross-

linking

Ampicillin

Penicillin antibioticCell wall synthesis inhibitor

Amino penicillinInhibits peptidoglycan cross-

linking

Anthraquinonescascara segrada, danthron, senna

Contact cathartics

Aprepitant dimenhydrinate

Antiemetic

Neurokinin 1 receptor antagonist

Atropine

Anticholinergic

AntimuscarinicTreatment for bradycardia,

diarrhea, cholinesterase poisoning

Azithromycin

Macrolide antibioticBacteriostatic protein synthesis

inhibitor

50S ribosome Inhibits translocation

Balsalazide

NSAID (salicylate)

Treatment of IBD

Bisacodyl

Contact cathartic

Bismuth subsalicylate

AntiulcerAntidiarrheal

Budesonide

AdrenocorticosteroidGlucocorticoid

Anti-inflammatory steroidInhaled OR treatment of IBD

Calcium carbonate

Antiulcer

Antacid

Cascara sagrada

Contact cathartic

Anthraquinone derivative

Castor Oil

Contact cathartic

Cimetidine

AntihistamineAntiulcer

H2 receptor antagonist

Cisapride

Prokinetic agent

5HT4 agonist

Clarithromycin

Macrolide antibioticBacteriostatic protein synthesis

inhibitor Antiulcer

50S ribosomeInhibits translocation

Danthron

Contact cathartic

Anthraquinone derivative

Dexamethasone

AdrenocorticosteroidGlucocorticoidAntineoplastic

Antiemetic

Anti-inflammatory steroidNot by inhalation

Dimenhydrinate

AntihistamineAntiemetic

H1 receptor antagonist

Diphenhydramine

Classical antihistamineAntiemetic

H1 antagonist

Diphenoxylate docusate

Antidiarrheal

Opiate

Docusates

Lubricating laxatives

Stool softeners

Doxycycline

Tetracycline antibioticBacteriostatic protein synthesis

inhibitor

30S ribosomePrevents aminoacyl tRNA attachment

Dronabinol

Antiemetic

Cannabinoid

Droperidol

Antiemetic

D2 receptor antagonist

Erythromycin

Macrolide antibioticBacteriostatic protein synthesis

inhibitor

50S ribosomeInhibits translocation

Granisetron

Antiemetic

5HT3 receptor antagonist

Infliximab

TNF inhibitor

Anti-TNF monoclonal antibody Treatment of IBD

Ipecac

Emetic

Kaolin

Antidiarrheal

Lactulose

Saline (osmotic) cathartic

Lansoprazole

Antiulcer

H+/K+ ATPase inhibitor

Loperamide

Antidiarrheal

Opiate

Magnesium hydroxide

AntiulcerSaline (osmotic) cathartic

Antacid

Meclizine

AntihistamineAntiemetic

H1 receptor antagonist

Mesalamine(5-ASA)

NSAID (salicylate)

Treatment of IBD

Methylcellulose

Bulk laxative

Metoclopramide

Prokinetic agentAntiemetic

D2 antagonist

Metronidazole

AntibioticAntiparasitic

Antiulcer

AnaerobesReduction leads to intermediates

that damage DNA

Mineral oil

Lubricating laxative

Stool softener

Minocycline

Tetracycline antibioticBacteriostatic protein synthesis

inhibitor

30S ribosomePrevents aminoacyl tRNA attachment

Misoprostol

ProstaglandinAntiulcer

Olsalazine

NSAID (salicylate)

Treatment of IBD

Omeprazole/esomeprazole

Antiulcer

H+/K+ ATPase inhibitor

Ondansetron

Antiemetic

5HT3 receptor antagonist

Oxytetracycline

Tetracycline antibioticBacteriostatic protein synthesis

inhibitor

30S ribosomePrevents aminoacyl tRNA attachment

Pantoprazole

Antiulcer

H+/K+ ATPase inhibitor

Pectin

Antidiarrheal

Polyethylene glycol- electolyte solution

AntidoteCathartic

Procarbazine

Antineoplastic

MiscellaneousProbably acts as alkylating

agent

Prochlorperazine

Antiemetic

D2 receptor antagonistPhenothiazine

Promethazine

Classical antihistamineAntipsychotic

Antiemetic

H1 antagonist

Rabeprazole

Antiulcer

H+/K+ ATPase inhibitor

Ranitidine

AntihistamineAntiulcer

H2 receptor antagonist

Rebamipide

Antiulcer

Senna

Contact cathartic

Anthraquinone derivative

Scopolamine

AnticholinergicAntiemetic

Muscarinic receptor antagonist

Simethicone

Anti-flatulent

Sodium bicarbonate

AntiulcerAntidote

AntacidAlkalinization of urine to treat drug toxicity (esp. barbiturates, salicylates,

methanol)

Sodium phosphate

Saline (osmotic) cathartic

Sucralfate

Antiulcer

Sulfasalazine

Disease modifyinganti-rheumatic drug (DMARD)

Metabolized to sulfonamide+ salicylate (NSAID) Treatment of IBD

Tegaserod

Antiemetic

5HT4 receptor agonist

Tetracycline

AntibioticBacteriostatic protein synthesis

inhibitor Antiulcer

30S ribosomePrevents aminoacyl tRNA attachment

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