novel 1,4-benzodiazepine-2,5-diones as hdm2 antagonists with improved cellular activity

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2006 Multi-membered N-heterocycles R 0690 Novel 1,4-Benzodiazepine-2,5-diones as Hdm2 Antagonists with Improved Cellu- lar Activity. — (LEONARD*, K.; et al.; Bioorg. Med. Chem. Lett. 16 (2006) 13, 3463-3468; Drug Discovery, Johnson & Johnson Pharm. Res. Dev., Exton, PA 19341, USA; Eng.) — M. Kowall 39- 194

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Page 1: Novel 1,4-Benzodiazepine-2,5-diones as Hdm2 Antagonists with Improved Cellular Activity

2006

200639.fm Seite 213 Freitag, 25. August 2006 12:00 12

Multi-membered N-heterocyclesR 0690 Novel 1,4-Benzodiazepine-2,5-diones as Hdm2 Antagonists with Improved Cellu-

lar Activity. — (LEONARD*, K.; et al.; Bioorg. Med. Chem. Lett. 16 (2006) 13, 3463-3468; Drug Discovery, Johnson & Johnson Pharm. Res. Dev., Exton, PA 19341, USA; Eng.) — M. Kowall

39- 194