Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

Invention Granted Under R.A. 8293 (PCT)

1 INVENTIONS

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2009/500117 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 13 January 2009

[54] Title: HUMANIZED ANTIBODY AGAINST AMYLOID BETA

[71] Proprietors(s): GENENTECH, INC., [US] and AC IMMUNE S.A. [CH]

[72] Inventor(s): ANDREA PFEIFER[CH]: MARIA PIHLGREN[CH]: ANDREAS MUHS[CH]: RYAN WATTS[US]

[73] Assignee(s): GENENTECH, INC., [US] and AC IMMUNE S.A. [CH]

[74] Attorney / Agent: E.B. ASTUDILLO AND ASSOCIATES

[30] Priority Data: 06014730.3 14/07/2006 EP; 06020765.1 02/10/2006 EP; 60/943,289 11/06/2007 US and 60/943,499 12/06/2007 US

[51] International Class 8: A 61P 25/28, C 07K 16/00, 16/18

[57] Abstract:

The present invention is related to chimeric and humanized antibody and to methods and compositions for the therapeutic and diagnostic use in the treatment of amyloidosis, a group of disorders and abnormalities associated with amyloid protein such as Alzheimer's disease.

Representative Drawing(s):

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[56] Reference(s) Cited and/or Considered:

Document description Document No.

BARD F ET AL: "Epitope and isotype specificities of antobodies to beta-amyloid peptide..." PROCEEDINGS OF THE NAT. ACAD. OF SCIEN. OF USA, NAT. ACAD. OF SCIE., WASH., DC, US, vol. 100, no. 4, 18 Feb. 2003, pg 2023-2028, XP002982464 ISSN: 0027-8424

1

LIU RUITIAN ET AL: "Single chain variable fragments against beta-amyloid (Abeta) can inhibit Abeta aggregation..." BIOCHEM., AMER. CHEM. SOC. EASTON, PA, US, vol. 43, no. 22, 12 May 2004, pg. 6959-6967, XP002395890 ISSN: 0006-2960

2

SOLOMON B ET AL: "MONOCLONAL ANTIBODIES INHIBIT IN VITRO... " PROCEEDINGS OF THE NAT. ACAD. OF SCIEN. OF USA, NAT. ACAD. OF SCIEN., WASH., DC, US, vol. 93, January 1996, pg 452-455, XP002942850 ISSN: 0027-8424

3

WO 2006/055178 A (MERCK & CO INC., ET AL.) 26 May 2006 4

WO 02/096937 A (NEUROCHEM INC, ET AL.) 5 DECEMBER 2002. 5

WO 03/070760 A (HOFFMANN LA ROCHE, ET AL.) 28 AUGUST 2003. 6

WO 00/72880 A (NEURALAB LTD, ET AL.) 7 DECEMBER 2000. 7

WO 01/62801 A (UNIV. WASHINGTON, ET AL.) 30 AUGUST 2001. 8

WO 2006/066171 A (NEURALAB LTD, ET AL.) 22 JUNE 2006. 9

No. of Claims: 600

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2009/500707 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 15 April 2009

[54] Title: CROPPING SYSTEMS FOR MANAGING WEEDS

[71] Proprietors(s): MONSANTO TECHNOLOGY LLC, [US]

[72] Inventor(s): CINDY ARNEVIK[US]: RONALD BRINKER[US]: GREG ELMORE[US]: JAMES GRAHAM[US]: ROBERT SAMMONS[US]: MICHELLE STARKE[US]: RICHARD VOTH[US]

[73] Assignee(s): MONSANTO TECHNOLOGY LLC, [US]

[74] Attorney / Agent: SYCIP SALAZAR HERNANDEZ AND GATMAITAN

[30] Priority Data: 11/758,660 05/06/2007 US and 60/862,907 25/10/2006 US

[51] International Class 8: A 01N 27/00, C 12N 15/82

[57] Abstract:

The invention provides cropping systems for managing weeds in crop environments. The cropping systems comprise, in one embodiment, transgenic plants that display tolerance to an auxin- like herbicide such as dicamba. Method for minimizing the development of herbicide resistant weeds were also provided.

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

NONE

No. of Claims: 46

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2011/500640 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 28 March 2011

[54] Title: NUTRITIONAL COMPOSITIONS LIPID GLOBULES WITH A CORE COMPRISING VEGETABLE LIPIDS AND A COATING COMPRISING PHOSPHOLIPIDS OR POLAR LIPIDS

[71] Proprietors(s): N.V. NUTRICIA [NL]

[72] Inventor(s): ANTOINE VAN BAALEN[NL]: ELINE MARLEEN VAN DER BEEK[NL]: CHRISTOPHER BEERMANN[DE]: GUNTHER BOEHM[DE]

[73] Assignee(s): N.V. NUTRICIA [NL]

[74] Attorney / Agent: HECHANOVA AND CO. INC.

[30] Priority Data: 08163478.4 02/09/2008 EP and 61/093,548 02/09/2008 US

[51] International Class 8: A 23L 1/29, 1/30

[57] Abstract:

The present invention relates to a nutritional composition for infants and/or toddlers comprising a lipid component which has a lipid globules coated with polar lipids. The composition can be used to prevent obesity and/or improve body composition later in life.

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

Document description Document No.

WO2006094995 (A1), ERDMANN PETER et al., 14 September 2006 (14.09.2006) 1

EP1800675 (A1), HAGEMAN ROBERT JOHAN JOSEPH et al., 27 June 2007 (27.06.2007) 2

WO2005051091 (A1), SHULMAN AVIDOR, 09 June 2005 (09.06.2005) 3

No. of Claims: 41

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2011/500949 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 17 May 2011

[54] Title: SOLID DOSAGE FORMS OF BENDAMUSTINE

[71] Proprietors(s): ASTELLAS DEUTSCHLAND GMBH [DE]

[72] Inventor(s): COLLEDGE, Jeff [NL]: PROFITLICH, Thomas Alfred [NL]: PATZAK, Ulrich[NL]: OUATAS, Taoufik[NL]: OLTHOFF, Margaretha[NL]

[73] Assignee(s): ASTELLAS DEUTSCHLAND GMBH [DE]

[74] Attorney / Agent: SIGUION REYNA MONTECILLO AND ONGSIAKO

[30] Priority Data: 08 020 996.8 03/12/2008 EP

[51] International Class 8: A 61K 31/4184, 9/20, 9/28

[57] Abstract:

In the present invention there is provided a pharmaceutical composition in a solid dosage form suitable for oral administration, the composition comprising bendamustine or a pharmaceutically acceptable ester, salt or solvate thereof as an active ingredient, and at least one pharmaceutically acceptable excipient, which is a pharmaceutically acceptable saccharide selected from the group consisting of one or more of a monosaccharide, a disaccharide, an oligosaccharide, a cyclic oligosaccharide, a polysaccharide and a saccharide alcohol, wherein the ratio by weight of the active ingredient to the saccharide excipient(s) is in the range of 1 :1-5.

Representative Drawing(s):

[56] Reference(s) Cited and/or Considered:

Document description Document No.

WO 2006/076620 A 20 July 2006 (20.07.2006) 1 US 2006/128777 A1 15 June 2006 (15.06.2006) 2

No. of Claims: 18

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2011/501298 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 22 June 2011

[54] Title: PLASMALOGEN COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND METHODS FOR TREATING DISEASES OF THE AGING

[71] Proprietors(s): PHENOMENOME DISCOVERIES, INC. [CA]

[72] Inventor(s): GOODENOWE, Dayan[CA]: WOOD, Paul, L. [CA]: AHIAHONU, Pearson [CA]: KHAN, Amin, M.[CA]: MANKIDY, Rishikesh[CA]

[73] Assignee(s): PHENOMENOME DISCOVERIES, INC. [CA]

[74] Attorney / Agent: CRUZ MARCELO & TENEFRANCIA

[30] Priority Data: 61/139,695 22/12/2008 US

[51] International Class 8: A 61K 31/232, 31/385, C 07C 227/02, 229/22, 319/02, 323/59, C 07D 339/04

[57] Abstract:

Described herein are routes of synthesis and therapeutic uses of 1-alkyl, 2-acyl glycerol derivatives of formula I: which when administered to mammalian biological systems result in increased cellular concentrations of specific sn-2 substituted ethanolamine plasmalogens independent of the ether lipid synthesis capacity of the system. Elevating levels of the specific sn-2 substituted species in this way can cause lowering of membrane cholesterol levels and the lowering of amyloid secretion.; These compounds can be used for the treatment or prevention of diseases of aging associated with increased membrane cholesterol, increased amyloid, and decreased plasmalogen levels, such as neurodegeneration (including Alzheimer's disease, Parkinson's disease and age-related macular degeneration), cognitive impairment, dementia, cancer (e.g. prostate, lung, breast, ovarian, and kidney cancers), osteoporosis, bipolar disorder and vascular diseases (such as atherosclerosis, hypercholesterolemia).

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

Document description Document No.

US 4,827,011 A May 1989 (05.1989) 1 US 5,759,585 A June 1998 (6.1998) 2

No. of Claims: 8

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2012/500646 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 29 March 2012

[54] Title: PHARMACEUTICAL COMPOSITION, PHARMACEUTICAL DOSAGE FORM, PROCESS FOR THEIR PREPARATION, METHODS FOR TREATING AND USES THEREOF

[71] Proprietors(s): BOEHRINGER INGELHEIM INTERNATIONAL GMBH [DE]

[72] Inventor(s): SCHNEIDER, PETER[DE]: EISENREICH, Wolfram[DE]: PEARNCHOB, NANTHARAT [DE]

[73] Assignee(s): BOEHRINGER INGELHEIM INTERNATIONAL GMBH [DE]

[74] Attorney / Agent: CASTILLO LAMAN TAN PANTALEON & SAN JOSE

[30] Priority Data: 09172081.3 02/10/2009 EP

[51] International Class 8: A 61K 31/155, 45/06, 47/02, 47/04, 47/10, 47/12, 47/14, 47/32, 47/36, 47/38, 47/42, 9/20, 9/28, 9/48, A 61P 13/12, 25/00, 27/12, 3/04, 3/08, 3/10, 43/00, 5/50, 9/00, 9/10

[57] Abstract: The present invention relates to pharmaceutical compositions comprising fixed dose combinations of a SGLT-2 inhibitor drug and a partner drug, processes for the preparation thereof, and their use to treat certain diseases.

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

Document description Document No.

WO 03099836 (04/12/2003) 1 WO 2007128761 (15/11/2007) 2 WO 2008055940 (15/05/2008) 3 WO 2008116179 (25/09/2008) 4 WO 2008101943 (28/08/2008) 5 Hussey, E. K. et. al.: "Safety, Pharmacokinetics and Pharmacodynamics of Remogliflozin Etabonate (SGLT2 Inhibitor) and Metformin When Co-Administered in Type 2 Diabetes Mellitus (T2DM) Patients" (DIABETES, AMERICAN DIABETES ASSOCIATION, US); 09/06/2009

6

No. of Claims: 19

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2012/501107 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 4 June 2012

[54] Title: DISSOLVABLE FILMS CONTAINING HIGH CONCENTRATIONS OF NONIONIC SURFACTANTS SUCH AS POLYSORBATES TO ENHANCE HIGH SOLID LOADINGS

[71] Proprietors(s): COLGATE-PALMOLIVE COMPANY [US]

[72] Inventor(s): MARTINETTI, Melissa[US]: JABBAL, Rajan[US]

[73] Assignee(s): COLGATE-PALMOLIVE COMPANY [US]

[74] Attorney / Agent: SYCIP SALAZAR HERNANDEZ AND GATMAITAN

[30] Priority Data: NONE

[51] International Class 8: A 61K 8/00, 8/02, A 61Q 11/00

[57] Abstract:

An oral care composition and method are described in which the composition includes a film or a plurality of film fragments entrained in a carrier. The film or plurality of film fragments comprises a relatively high concentration of nonionic surfactants. The composition and methods provide benefits including higher active material loading in the film formula for improved efficacy, and a reduced amount of film needed in a product, which at the same time delivering comparable or improved efficacy with lower loading of the film in the composition.

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

Document description Document No.

US2005106112 (A1) , BOYD THOMAS J. et al., 19 May 2005 (19.05.2005) 1

US5948430 (A), ZERBE HORST GEORG et al., 07 September 1999 (07.09.1999) 2

US6231957 (B1), ZERBE HORST G et al., 15 May 2001 (15.05.2001) 3

No. of Claims: 13

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2012/502183 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 6 November 2012

[54] Title: CARBOHYDRATE POLYAMINE BINDERS AND MATERIALS MADE THEREWITH

[71] Proprietors(s): KNAUF INSULATION [BE]

[72] Inventor(s): APPLEY, Charles[US]: HAMPSON, Carl[GB]: MUELLER, Gert[DE]: PACOREL, Bénédicte[FR]

[73] Assignee(s): KNAUF INSULATION [BE]

[74] Attorney / Agent: AGCAOILI & ASSOCIATES

[30] Priority Data: 61/332,458 07/05/2010 US

[51] International Class 8: C 08G 12/00, 14/00, 16/00

[57] Abstract:

A binder comprising the products of a carbohydrate reactant and polyamine is disclosed. The binder is useful for consolidating loosely assembled matter, such as fibers. Uncured fibrous products comprising fibers in contact with a carbohydrate reactant and a polyamine are also disclosed. The binder composition may be cured to yield a fibrous product comprising fibers bound by a cross-linked polymer. Further disclosed are methods for binding fibers with the carbohydrate reactant and polyamine based binder.

Representative Drawing(s):

[56] Reference(s) Cited and/or Considered:

Document description Document No.

US 2 198 874 A (LEIGHTON HOLMES ERIC) 30 April 1940 1 US 2 442 989 A (SIDNEY SUSSMAN) 8 June 1948 2 US 4 085 076 (GIBBONS JOHN, ET AL) 18 April 1978 3

No. of Claims: 27

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2013/500096 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 14 January 2013

[54] Title: REDISPERSIBLE DRY COMPOSITION OF POLYMER FINISHES OR OTHER PRODUCTS FOR THE CONSTRUCTION

[71] Proprietors(s): PAREXGROUP SA [FR]

[72] Inventor(s): DANTIN, Véronique[FR]: LEPLEY, Gérard[FR]: GONCALO, Paulo[FR]: NONES, Carlos[US]: PAREDES, Pedro[US]

[73] Assignee(s): PAREXGROUP SA [FR]

[74] Attorney / Agent: HECHANOVA & CO., INC.

[30] Priority Data: PCT/EP2010/060337 16/07/2010 EP

[51] International Class 8: C 04B 26/02, 26/04, 26/06, 28/06, 28/16, C 09D 5/03

[57] Abstract:

The invention relates to improved non-efflorescing cement-free and water-dispersible powder building material compositions comprising a homopolymer or copolymer as binder, useful for the preparation of wet formulations of plasters grouts, waterproofing coatings or mortars for the construction and the civil engineering industry. Redispersible dry composition of polymer finish comprising: a powdery organic binder included a polymer obtained by spray-drying or lyophilisation of a dispersion containing said polymer and a protective colloid; a deprotection agent; a specific adsorbent filler; and/or a load; and/or a water retentive agent; and/or a mineral rheological agent; and/or a defoamer; and/or a biocide; and/or a pigment. The invention also refers to the methods of preparation of these dry compositions and wet formulations, the application of these latter onto the surface of buildings or civil engineering works, the so obtained coatings as well as the so coated elements. The applications of these wet formulations can be also hardened joints or other hardened products for the construction as well as hardened mass objects. All these hardened products are remarkably water-resistant, non efflorescent and easy to obtain.

Representative Drawing(s):

[56] Reference(s) Cited and/or Considered:

Document description Document No.

CN 101 481 584 A (Univ. Soutj China Tech.) 15 July 2009 1 DE 199 10 602 C1 (Wacker Chemie GMBH) 16 November 2000 2

JP 2006 335597 A (Saeki KK) 14 December 2006 3 US 3 867 335 (Reed Delmer et al) 18 February 1975 4 EP 1 593 721 (Wacker Polymer Systems GMBH) 9 5

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

November 2005

No. of Claims: 84

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2013/502118 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 11 October 2013

[54] Title: ARYL-OR HETEROARYL-SUBSTITUTED BENZENE COMPOUNDS

[71] Proprietors(s): EPIZYME, INC. [US]

[72] Inventor(s):

KUNTZ, Kevin Wayne[US]: CHESWORTH, Richard[GB]: DUNCAN, Kenneth William[GB]: KEILHACK, Heike[DE]: WARHOLIC, Natalie[US]: KLAUS, Christine[US]: SEKI, Masashi[JP]: SHIROTORI, Syuji[JP]: KAWANO, Satoshi[JP]: WIGLE, Timothy James Nelson[US]

[73] Assignee(s): EPIZYME, INC. [US]

[74] Attorney / Agent: E. B. ASTUDILLO & ASSOCIATES

[30] Priority Data: 61/474,821 13/04/2011 US and 61/499,595 21/06/2011 US

[51] International Class 8: A 61K 31/435, 31/4433, 31/4439, 31/444, 31/4545, 31/4709, 31/496, 31/506, 31/5377, 31/551, 31/553, A 61P 35/00, C 07D 213/64, 401/12, 401/14, 405/12, 405/14, 409/12, 413/12, 413/14, 417/12, 491/08, 491/107

[57] Abstract:

The present invention relates to aryl- or heteroaryl-substituted benzene compounds. The present invention also relates to pharmaceutical compositions containing these compounds and methods of treating cancer by administering these compounds and pharmaceutical compositions to subjects in need thereof. The present invention also relates to the use of such compounds for research or other non-therapeutic purposes.

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

Document description Document No.

US 2005266473 (01/12/2005) 1 US 4522811 (11/06/1985) 2 US 5763263 (09/06/1998) 3

No. of Claims: 314

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2013/502319 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 12 November 2013

[54] Title: PYRROLIDINYL UREA, PYRROLIDINYL THIOUREA AND PYRROLIDINYL GUANIDINE COMPOUNDS AS TRKA KINASE INHIBITORS

[71] Proprietors(s): ARRAY BIOPHARMA INC. [US]

[72] Inventor(s):

ALLEN, Shelley[GB]: ANDREWS, Steven, W.[US]: BLAKE, James, F.[US]: CONDROSKI, Kevin, R.[US]: HAAS, Julia[US]: HUANG, Lily[US]: JIANG, Yutong[US]: KERCHER, Timothy[US]: KOLAKOWSKI, Gabrielle R.[US]: SEO, Jeongbeob[US]

[73] Assignee(s): ARRAY BIOPHARMA INC. [US]

[74] Attorney / Agent: BUCOY POBLADOR & ASSOCIATES

[30] Priority Data: 61/485,858 13/05/2011 US

[51] International Class 8: A 61K 31/4155, 31/4162, 31/4178, 31/4192, C 07D 401/14, 403/12, 403/14, 405/14, 409/14, 413/14, 417/14, 471/04, 487/04, 491/04, 495/04

[57] Abstract:

Compounds of Formula I: or stereoisomers, tautomers, or pharmaceutically acceptable salts, or solvates or prodrugs thereof, where R

1, R

2, R

a, R

b, R

c, R

d,

X, Y, B, and Ring C are as defined herein, and wherein the Y-B moiety and the NH-C(=X)-NH moiety are in the trans configuration, are inhibitors of TrkA kinase and are useful in the treatment of diseases which can be treated with a TrkA kinase inhibitor such as pain, cancer, inflammation, neurodegenerative diseases and certain infectious diseases.

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

Document description Document No.

WO 2010/048314 A1 29 April 2010 (29.04.2010) 1 WO 99/32110 A1 01 July 1999 (01.07.1999) 2 WO 2010/040663 A1 15 April 2010 (15.04.2010) 3 JP 2005 206527 A 04 August 2005 (04.08.2005) 4

No. of Claims: 768

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2013/502434 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 22 November 2013

[54] Title: SUBSTITUTED PYRIDOPYRAZINES AS NOVEL SYK INHIBITORS

[71] Proprietors(s): HUTCHISON MEDIPHARMA LIMITED [CN]

[72] Inventor(s): SU, Wei-Guo[US]: DENG, Wei[CN]: JI, Jianguo[US]

[73] Assignee(s): HUTCHISON MEDIPHARMA LIMITED [CN]

[74] Attorney / Agent: CRUZ MARCELO & TENEFRANCIA

[30] Priority Data: PCT/CN2011/075431 08/06/2011 CN

[51] International Class 8: A 61K 31/4985, 31/5377, 31/541, 31/551, 31/553, A 61P 11/02, 19/02, 25/00, 29/00, 35/00, 35/02, 37/02, 37/08, 43/00, 7/00, 7/06, C 07D 471/04, 519/00

[57] Abstract: Provided are pyridopyrazine compounds of formula (I), pharmaceutical compositions thereof and methods of use therefore, wherein R1, R2, R3, R4 and m are as defined in the specification.

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

Document description Document No.

WO 2004/005472 (15/01/2004) 1 CARROLL TEMPLE, JR. ET AL., "1,2-Dihydropyrido[3,4-b] pyrazines: Structure-Activity Relationships.", J. MED. CHEM., (1983)

2

JEFFREY W. WILLIAMS ET AL., "The inhibition of dihydrofolate reductase by folate analogues: structural requirements for slow- and tight-binding inhibition.", BIOCHEMICAL PHARMACOLOGY, (1980)

3

BRITTA NISIUS ET AL., "Development of a Fingerprint Reduction Approach for Bayesian Similarity Searching Based on Kullback-Leibler Divergence Analysis.", J. CHEM. INF. MODEL., (2009)

4

ROBERT D. ELLIOTT ET AL., "Potential Folic Acid Antagonists. VI. The Syntheses of 1- and 3-Deazamethotrexate.", J. ORG. CHEM., (1971)

5

No. of Claims: 34

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2013/502583 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 11 December 2013

[54] Title: METHOD AND SYSTEM FOR PROCESSING IMAGE DATA OBTAINED FROM SCANNING A NETWORK INFRASTRUCTURE

[71] Proprietors(s): Fugro ROAMES Pty Ltd. [AU]

[72] Inventor(s): BANGAY, James Gordon[AU]

[73] Assignee(s): Fugro ROAMES Pty Ltd. [AU]

[74] Attorney / Agent: CASTILLO LAMAN TAN PANTALEON & SAN JOSE

[30] Priority Data: 2011901865 16/05/2011 AU

[51] International Class 8: G 06K 9/00, G 06T 7/00

[57] Abstract:

The invention relates to a method and system for processing image data obtained from scanning a network infrastructure for the detection and analysis of specific objects of interest, such as powerlines and other overhead conductors, or similar structures. The image data comprises a plurality of co-ordinate points in three-dimensional space, and in order to identify conductors in the network infrastructure, the method involves analysing the co-ordinate points to identify sets of co-ordinate points indicative of a set of substantially parallel lines, and analysing the co¬ ordinate points on the basis of said identified substantially parallel lines thereby to allow identification and mapping of hanging catenaries representing said conductors.

Representative Drawing(s):

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[56] Reference(s) Cited and/or Considered:

Document description Document No.

US 9,384,399 B2 / Dow, et al. / 16 May 2006 1 WO 2011/088509 A1 / JRB Engineering Pty Ltd. / 28 July 2011 2

No. of Claims: 33

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2014/502403 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 27 October 2014

[54] Title: PAINT BOOTH WITH PURIFIER

[71] Proprietors(s): BUNRI INCORPORATION [JP]

[72] Inventor(s): TASHIRO, Makoto[JP]: TASHIRO, Minoru[JP]

[73] Assignee(s): BUNRI INCORPORATION [JP]

[74] Attorney / Agent: SAPALO VELEZ BUNDANG & BULILAN LAW OFFICES

[30] Priority Data: 2013-121197 07/06/2013 JP

[51] International Class 8: B 05B 1/14, 15/04, 15/12

[57] Abstract:

A paint booth (10) is provided with a booth body (12) and a purifier (13). The purifier (13) is provided with a water tank (20), water rope formation mechanism (22), sludge removal mechanism (26), exhaust mechanism (28), barrier member (45), inclined plate (50), and windshield plate (60). Water falling from nozzles (35) of a water case (30) forms a large number of water ropes (40). The inclined plate (50) has a water receiving surface (55) sloping forwardly down at an angle (8) from a vertically intermediate part (H3) of the barrier member (45) toward a water surface (W1) of the water tank (20). A lower end (62) of the windshield plate (60) is in contact with water (W) in the water tank (20). An airflow reversal section (53) is formed between a lower end (52) of the inclined plate (50) and the water surface (W1). Air directed downward from an airflow inlet (59) is turned upward at the airflow reversal section (53) and directed to an exhaust chamber (46) through air circulation sections (65, 66).

Representative Drawing(s):

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[56] Reference(s) Cited and/or Considered:

Document description Document No.

EP 2 409 779 A1, BUNRI INC, Paint booth equipped with purification device, 25 January 2012 1

GB1004239 A, TUNZINI, Improvements in or relating to removal of suspended matter from gases, 15 September 1965

2

No. of Claims: 19

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2015/500068 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 12 January 2015

[54] Title: MODULAR BUILDING

[71] Proprietors(s): 1 SPACE PTY LTD [AU]

[72] Inventor(s): UNGER, Susan[AU]

[73] Assignee(s): 1 SPACE PTY LTD [AU]

[74] Attorney / Agent: VILLARAZA & ANGANGCO

[30] Priority Data: 2012902966 11/07/2012 AU; 2013100359 24/03/2013 AU; 2013201852 24/03/2013 AU; 2013900027 04/01/2013 AU; 2013900029 04/01/2013 AU and 2013900962 19/03/2013 AU

[51] International Class 8: E 04B 1/343, 1/348, E 04H 1/02

[57] Abstract:

A modular building unit for construction of a building comprises a structural frame 40 suitable for interconnection to another modular building unit in construction of the building; and a stud frame wall 80/82 internal to and fixed to the frame. The modular building unit is suitable for handling as a shipping container for transport.

Representative Drawing(s):

[56] Reference(s) Cited and/or Considered:

Document description Document No.

WO 2008/027234 A1 ABRAMS, Alexander et al. 06 March 2008 (06.03.2008) 1

US 5 511 908 B1 VAN, Norman et al. 30 April 1996 (30.04.1996) 2

No. of Claims: 33

Intellectual Property Center, 28 Upper McKinley Rd. McKinley Hill Town Center, Fort Bonifacio, Taguig City 1634 Philippines

Tel. No. 238-6300 Website: http://www.ipophil.gov.ph e-mail: mail@ipophil.gov.ph

Volume 20 Number 68 Date Released: June 23, 2017

[19] INTELLECTUAL PROPERTY PHILIPPINES

[12] INVENTION GRANT

[21] Registration Number: 1/2015/500373 Document Code: B1

[45] Issue Date: 31 March 2017

[22] Date Filed: 20 February 2015

[54] Title: DIAZEPINONE DERIVATIVES USEFUL FOR THE TREATMENT OF FRAGILE X SYNDROME, PARKINSONS OR REFLUX DISEASE

[71] Proprietors(s): NOVARTIS AG [CH]

[72] Inventor(s): BEHNKE, Dirk[DE]: CARCACHE, David[CH]: ERTL, Peter[CH]: KOLLER, Manuel[CH]: ORAIN, David[FR]

[73] Assignee(s): NOVARTIS AG [CH]

[74] Attorney / Agent: E.B. ASTUDILLO & ASSOCIATES

[30] Priority Data: 1215033.0 23/08/2012 GB

[51] International Class 8: A 61K 31/551, A 61P 1/04, 25/16, 25/28, C 07D 471/04

[57] Abstract:

The invention relates to compound of the formula I

or a salt thereof, wherein the substituents are as defined in the specification; to its preparation, to its use as medicament and to medicaments comprising it.

Representative Drawing(s): NONE

[56] Reference(s) Cited and/or Considered:

Document description Document No.

WO 2004/087048 A2 (MERCK & CO INC [US]) 14 October 2004 1

No. of Claims: 251